某些化学实体、组合物及方法_2

文档序号:8490840阅读:来源:国知局
6-羰基)苯基)丙烷-1-磺酰胺, N-(3-氟-5-(吡啶并[3, 4-b]吡嗪-7-羰基)苯基)丙烷-1-磺酰胺, (3-氟-5-(1,5-萘啶-2-羰基)苯基)丙烷-1-磺酰胺, N-(3-(苯并[d]噁唑-6-羰基)-5-氟苯基)丙烷-1-磺酰胺, N-(3-(苯并[d]噁唑-5-羰基)-5-氟苯基)丙烷-1-磺酰胺, N-(3-氟-5-(噁唑并[5, 4-b]吡啶-5-羰基)苯基)丙烷-1-磺酰胺, N- (3-(苯并[d]噻唑-6-羰基)-5-氟苯基)丙烷-1-磺酰胺, N-(3-(3a,7a-二氢-1H-吡唑并[3, 4-b]吡啶-3-羰基)-5-氟苯基)丙烷-1-磺酰 胺, N-(3-(7, 7a-二氢-4aH-吡咯并[2, 3-d]嘧啶-5-羰基)-5-氟苯基)丙烷-1-磺酰 胺, N-(3-(5, 7a-二氢-4aH-吡咯并[2, 3-b]吡嗪-7-羰基)-5-氟苯基)丙烷-1-磺酰 胺, N-(3-(3a,7a-二氢-1H-吡唑并[3, 4-b]吡嗪-3-羰基)-5-氟苯基)丙烷-1-磺酰 胺, N-(3-(7, 7a-二氢-4aH-吡咯并[2, 3-c]哒嗪-5-羰基)-5-氟苯基)丙烷-1-磺酰 胺, N-(3-氟_5_ (3-((2-羟基乙基)氨基)喹啉_6_幾基)苯基)丙烷-1-横酰胺, N- (3-氟-5- (3-(吡咯烷-1-基)喹啉-6-羰基)苯基)丙烷-1-磺酰胺, N-(3-(3-(1H-咪唑-1-基)喹啉-6-羰基)-5-氟苯基)丙烷-1-磺酰胺, N- (3- (3- (1H-吡唑-4-基)喹啉-6-羰基)-5-氟苯基)丙烷-1-磺酰胺, N-(2, 5-二氟_3_ (喹啉_6_幾基)苯基)丙烷-1-横酰胺, N-(2, 5-二氟-3-(3-甲基喹啉-6-羰基)苯基)丙烷-1-磺酰胺, N-(3-(3-氛基喹啉_6_幾基)-2, 5-二氟苯基)丙烷-1-横酰胺, N-(2, 5-二氟-3-(3-甲氧基喹啉-6-羰基)苯基)丙烷-1-磺酰胺, N-(3-(3-(4-氯苯基)喹啉_6_幾基)-2, 5-二氟苯基)丙烷-1-横酰胺, N- (2, 5-二氟_3_ (3- (P比啶_3_基)喹啉_6_幾基)苯基)丙烷-1-横酰胺, N-(2, 5-二氟-3-(3-吗啉基喹啉-6-羰基)苯基)丙烷-1-磺酰胺, N-(2, 5-二氟-3-(3-(哌嗪-1-基)喹啉-6-羰基)苯基)丙烷-1-磺酰胺, N-(2, 5-二氟_3_(3-(2-羟基乙氧基)喹啉_6_幾基)苯基)丙烷-1-横酰胺, N- (2, 5-二氟-3-(喹唑啉-6-羰基)苯基)丙烷-1-磺酰胺, N-(2, 5-二氟-3-(1,7-萘啶-6-羰基)苯基)丙烷-1-磺酰胺, N-(2, 5-二氟-3-(P比啶并[3, 4_b]P比嘆-7-羰基)苯基)丙烷-1-磺酰胺, N-(2, 5-二氟_3_ (1,5-萘啶_2_幾基)苯基)丙烷-1-横酰胺, N- (3-(苯并[d]噁唑-6-羰基)-2, 5-二氟苯基)丙烷-1-磺酰胺, N-(3-(苯并[d]噁唑-5-羰基)-2, 5-二氟苯基)丙烷-1-磺酰胺, N-(2, 5-二氟-3-(噁唑并[5, 4-b]吡啶-5-羰基)苯基)丙烷-1-磺酰胺, N-(3-(苯并[d]噻唑-6-羰基)-2, 5-二氟苯基)丙烷-1-磺酰胺, N_ (3_ (3a, 7a_二氛-1H-吡挫并[3, 4_b]吡啶_3_幾基)_2, 5_二氣苯基)丙烷_1_横 酰胺, N-(3-(7, 7a_二氢_4aH_P比略并[2, 3_d]喃啶_5_幾基)-2, 5-二氟苯基)丙烷-1-横 酰胺, N-(3-(5, 7a_二氢_4aH_P比略并[2, 3_b]P比嘆_7_幾基)-2, 5-二氟苯基)丙烷-1-横 酰胺, N_ (3_ (3a, 7a_二氛-1H-吡挫并[3, 4_b]吡嘆_3_幾基)_2, 5_二氣苯基)丙烷_1_横 酰胺, N-(3-(7, 7a_ 二氢 _4aH_P比略并[2, 3_c] _嘆 _5_ 幾基)-2, 5-二氟苯基)丙烷-1-横 酰胺, N-(2, 5-二氟_3_ (3-((2-羟基乙基)氨基)喹啉_6_幾基)苯基)丙烷-1-横酰胺,N-(2, 5-二氟_3_ (3-(P比略烧-1-基)喹啉_6_幾基)苯基)丙烷-1-横酰胺, N-(3-(3-(1H-咪唑-1-基)喹啉-6-羰基)-2, 5-二氟苯基)丙烷-1-磺酰胺, N- (3- (3- (1H-吡唑-4-基)喹啉-6-羰基)-2, 5-二氟苯基)丙烷-1-磺酰胺, N- (3, 4-二氟-5-(喹啉-6-羰基)苯基)丙烷-1-磺酰胺, N-(3, 4-二氟-5-(3-甲基喹啉-6-羰基)苯基)丙烷-1-磺酰胺, N-(3-(3-氰基喹啉-6-羰基)-4, 5-二氟苯基)丙烷-1-磺酰胺, N-(3, 4-二氟-5-(3-甲氧基喹啉-6-羰基)苯基)丙烷-1-磺酰胺, N-(3-(3-(4-氯苯基)喹啉-6-羰基)-4, 5-二氟苯基)丙烷-1-磺酰胺, N- (3, 4-二氟-5- (3-(吡啶-3-基)喹啉-6-羰基)苯基)丙烷-1-磺酰胺, N-(3, 4-二氟-5-(3-吗啉基喹啉-6-羰基)苯基)丙烷-1-磺酰胺, N-(3, 4-二氟-5-(3-(哌嗪-1-基)喹啉-6-羰基)苯基)丙烷-1-磺酰胺, N-(3, 4-二氟-5-(3-(2-羟基乙氧基)喹啉-6-羰基)苯基)丙烷-1-磺酰胺, N- (3, 4-二氟-5-(喹唑啉-6-羰基)苯基)丙烷-1-磺酰胺, N-(3, 4-二氟-5-(1,7-萘啶-6-羰基)苯基)丙烷-1-磺酰胺, N-(3, 4-二氟-5-(吡啶并[3, 4-b]吡嗪-7-羰基)苯基)丙烷-1-磺酰胺, N-(3, 4-二氟-5-(1,5-萘啶-2-羰基)苯基)丙烷-1-磺酰胺, N- (3-(苯并[d]噁唑-6-羰基)-4, 5-二氟苯基)丙烷-1-磺酰胺, N- (3-(苯并[d]噁唑-5-羰基)-4, 5-二氟苯基)丙烷-1-磺酰胺, N-(3, 4-二氟-5-(噁唑并[5, 4-b]吡啶-5-羰基)苯基)丙烷-1-磺酰胺, N-(3-(苯并[d]噻唑-6-羰基)-4, 5-二氟苯基)丙烷-1-磺酰胺, N_ (3_ (3a, 7a_二氛-1H-吡挫并[3, 4_b]吡啶_3_幾基)_4, 5_二氣苯基)丙烷_1_横 酰胺, N- (3- (7, 7a-二氢-4aH-吡咯并[2, 3-d]嘧啶-5-羰基)-4, 5-二氟苯基)丙烷-1-磺 酰胺, N- (3- (5, 7a-二氢-4aH-吡咯并[2, 3-b]吡嗪-7-羰基)-4, 5-二氟苯基)丙烷-1-磺 酰胺, N- (3- (3a,7a-二氢-1H-吡唑并[3, 4-b]吡嗪-3-羰基)-4, 5-二氟苯基)丙烷-1-磺 酰胺, N- (3- (7, 7a-二氢-4aH-吡咯并[2, 3-c]哒嗪-5-羰基)-4, 5-二氟苯基)丙烷-1-磺 酰胺, N-(3, 4-二氟_5_ (3-((2-羟基乙基)氨基)喹啉_6_幾基)苯基)丙烷-1-横酰胺,N- (3, 4-二氟-5- (3-(吡咯烷-1-基)喹啉-6-羰基)苯基)丙烷-1-磺酰胺, N-(3-(3-(1H-咪唑-1-基)喹啉-6-羰基)-4, 5-二氟苯基)丙烷-1-磺酰胺, N- (3- (3- (1H-吡唑-4-基)喹啉-6-羰基)-4, 5-二氟苯基)丙烷-1-磺酰胺, N- (2, 4, 5-三氟-3-(喹啉-6-羰基)苯基)丙烷-1-磺酰胺, N-(2, 4, 5-三氟-3-(3-甲基喹啉-6-羰基)苯基)丙烷-1-磺酰胺, N-(3-(3-氰基喹啉-6-羰基)-2, 4, 5-三氟苯基)丙烷-1-磺酰胺, N-(2, 4, 5-三氟-3-(3-甲氧基喹啉-6-羰基)苯基)丙烷-1-磺酰胺, N-(3-(3-(4-氯苯基)喹啉-6-羰基)-2, 4, 5-三氟苯基)丙烷-1-磺酰胺, N- (2, 4, 5-三氟-3- (3-(吡啶-3-基)喹啉-6-羰基)苯基)丙烷-1-磺酰胺, N-(2, 4, 5-三氟-3-(3-吗啉基喹啉-6-羰基)苯基)丙烷-1-磺酰胺, N-(2, 4, 5-三氟-3-(3-(哌嗪-1-基)喹啉-6-羰基)苯基)丙烷-1-磺酰胺, N-(2, 4, 5-三氟-3-(3-(2-羟基乙氧基)喹啉-6-羰基)苯基)丙烷-1-磺酰胺, N- (2, 4, 5-三氟-3-(喹唑啉-6-羰基)苯基)丙烷-1-磺酰胺, N-(2, 4, 5-三氟-3-(1,7-萘啶-6-羰基)苯基)丙烷-1-磺酰胺, N-(2, 4, 5-三氟-3-(吡啶并[3, 4-b]吡嗪-7-羰基)苯基)丙烷-1-磺酰胺, N-(2, 4, 5-二氟-3-(1,5-萘啶-2-羰基)苯基)丙烷-1-磺酰胺, N-(3-(苯并[d]噁唑-6-羰基)-2, 4, 5-三氟苯基)丙烷-1-磺酰胺, N-(3-(苯并[d]噁唑-5-羰基)-2, 4, 5-三氟苯基)丙烷-1-磺酰胺, N-(2, 4, 5-三氟-3-(噁唑并[5, 4-b]吡啶-5-羰基)苯基)丙烷-1-磺酰胺, N-(3-(苯并[d]噻唑-6-羰基)-2, 4, 5-三氟苯基)丙烷-1-磺酰胺, N- (3- (3a, 7a~ 一氛_1H-吡挫并[3, 4-b]吡陡幾基)-2, 4, 5-二氣苯基)丙烷横 酰胺, N-(3-(7,7a-二氢-4aH-吡咯并[2,3-d]嘧啶-5-羰基)-2,4,5_三氟苯基)丙烷-1-磺 酰胺, ^(3-(5,7&-二氢-4&11-吡咯并[2,3-13]吡嗪-7-羰基)-2,4,5-三氟苯基)丙烷-1-磺 酰胺, N-(3-(3a,7a-二氢-1H-吡唑并[3, 4-b]吡嗪-3-羰基)-2, 4, 5-三氟苯基)丙烷-1-磺 酰胺, ^(3-(7,7&-二氢-4&11-吡咯并[2,3-(3]哒嗪-5-羰基)-2,4,5-三氟苯基)丙烷-1-磺 酰胺, N-(2, 4, 5-二氟_3_ (3-((2-羟基乙基)氨基)喹啉_6_幾基)苯基)丙烷-1-横酰 胺, N- (2, 4, 5-三氟-3- (3-(吡咯烷-1-基)喹啉-6-羰基)苯基)丙烷-1-磺酰胺, N-(3-(3-(1H-咪唑-1-基)喹啉-6-羰基)-2, 4, 5-三氟苯基)丙烷-1-磺酰胺, N- (3- (3- (1H-吡唑-4-基)喹啉-6-羰基)-2, 4, 5-三氟苯基)丙烷-1-磺酰胺, 1_ (3-氟-5_ (喹啉_6_幾基)苯基)_3_ (3-氟苯基)脈, 1_ (3-氟-5_ (3-甲基喹啉_6_幾基)苯基)_3_ (3-氟苯基)脈, 1- (3- (3-氛基喹啉_6_幾基)_5_氟苯基)_3_ (3-氟苯基)脈, 1_ (3-氟-5_ (3-甲氧基喹啉_6_幾基)苯基)_3_ (3-氟苯基)脈, 1_ (3-氣-5- (3_吗琳基卩奎琳_6_幾基)苯基)_3_ (3_氣苯基)脈, I- (3, 4_二氣苯基)_3_ (3_氣_5_ (3_吗琳基卩奎琳_6_幾基)苯基)脈, 1- (3-氟-5- (3-吗啉基喹啉-6-羰基)苯基)-3- (4-氟苯基)脲, 1_ (4-氣苯基)-3_ (3_氣_5_ (3_吗琳基卩奎琳_6_幾基)苯基)脈, 1_ (3-氣苯基)-3_ (3_氣_5_ (3_吗琳基卩奎琳_6_幾基)苯基)脈, 1-(4-氯-3-(三氟甲基)苯基)-3-(3-氟-5-(3-吗啉基喹啉-6-羰基)苯基)脲, 1_ (3-氟-5_ (3- (B比略烧-1-基)喹啉_6_幾基)苯基)_3_ (3-氟苯基)脈, 1- (3-氟-5- (3-(哌嗪-1-基)喹啉-6-羰基)苯基)-3- (3-氟苯基)脲, 1- (3, 4-二氟苯基)-3- (3-氟-5- (3-(哌嗪-1-基)喹啉-6-羰基)苯基)脲, 1- (3-氟-5- (3-(哌嗪-1-基)喹啉-6-羰基)苯基)-3- (4-氟苯基)脲, 1- (4-氯苯基)-3- (3-氟-5- (3-(哌嗪-1-基)喹啉-6-羰基)苯基)脲, 1- (3-氟_5_ (3-(啦啶_3_基)喹卩林_6_幾基)苯基)_3_ (3-氟苯基)脈, 1-(3-氟_5_ (3-((2-羟基乙基)氨基)喹卩林_6_幾基)苯基)_3_ (3-氟苯基)脈, I-(3_氣_5_ (3_ (2_羟基乙氧基)卩奎卩林_6_幾基)苯基)_3_ (3_氣苯基)脈, 1- (3- (3- (1H-吡唑-4-基)喹啉-6-羰基)-5-氟苯基)-3- (3-氟苯基)脲, 1- (3- (3- (1H-咪唑-1-基)喹啉-6-羰基)-5-氟苯基)-3- (3-氟苯基)脲, I- (3_氣_5_ (卩奎挫卩林_6_幾基)苯基)_3_ (3_氣苯基)脈, 1- (3-氟-5-(喹唑啉-6-羰基)苯基)-3- (4-氟苯基)脲, I- (3, 4_二氣苯基)_3_ (3_氣_5_ (卩奎挫卩林_6_幾基)苯基)脈, 1- (3-氟_5_ (1,7-萘啶_6_幾基)苯基)_3_ (3-氟苯基)脈, 1- (3, 4-二氟苯基)_3_ (3-氟_5_ (1,7-萘啶_6_幾基)苯基)脈, 1- (3-氟_5_ (3-吗卩林基-1,7-萘啶_6_幾基)苯基)_3_ (3-氟苯基)脈, 1- (3, 4-二氟苯基)_3_ (3-氟_5_ (3-吗卩林基-1,7-萘啶_6_幾基)苯基)脈, 1- (3-氟_5_ (啦啶并[3, 4_b]啦嗪_7_幾基)苯基)_3_ (3-氟苯基)脈, 1- (3-氟_5_ (啦啶并[3, 4_b]啦嗪_7_幾基)苯基)_3_ (4-氟苯基)脈, 1-(3-氟-5-(2-吗啉基吡啶并[3, 4-b]吡嗪-7-羰基)苯基)-3-(4-氟苯基)脲, 1-(3-氟_5_ (2-吗卩林基啦啶并[3, 4_b]啦嗪_7_幾基)苯基)_3_ (3-氟苯基)脈, 1- (3-氟_5_ (1,5-萘啶_2_幾基)苯基)_3_ (3-氟苯基)脈, 1- (3-氟_5_ (7-吗卩林基-1,5-萘啶_2_幾基)苯基)_3_ (3-氟苯基)脈, 1- (3_ (苯并[d]D惡挫_6_幾基)_5_氟苯基)_3_ (3_氟
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